Description
PROTAC ERalpha Degrader-2 comprises a cIAP1 ligand binding group, a linker and an estrogen receptor alpha (ERalpha) binding group. PROTAC ERalpha Degrader-2 is an ERalpha degrader. Maximal ERalpha degradation at 30uM concentration in Human mammary tumor MCF7 cells. Degradation inducers based on cIAP1 are called specific and non-genetic IAP-dependent protein erasers (SNIPERs)[1]